SCHEMBL9544449

SCHEMBL9544449

COC(=O)COc1ccc(CCN(CC(O)c2cccc(Br)c2)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 8/20 0.43
ADRB1 P08588 5/20 0.43
ADRB2 P07550 2/20 0.43
GLA P06280 1/20 0.43
BACE1 P56817 6/20 0.41
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
FFAR1 O14842 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9544456 1.00 ADRB3 (0.43) ADRB3ADRB1ADRB2GLABACE1
SCHEMBL9543347 0.89 MEN1 (0.44) ADRB3ADRB1ADRB2GLABACE1
SCHEMBL9543338 0.89 MEN1 (0.44) ADRB3ADRB1ADRB2GLABACE1
SCHEMBL9545127 0.79 LTB4R2 (0.44) ADRB3ADRB1ADRB2BACE1FFAR1
SCHEMBL4462454 0.79 BACE1 (0.43) ADRB3ADRB1ADRB2BACE1
SCHEMBL1622477 0.79 BACE1 (0.43) ADRB3ADRB1ADRB2BACE1
SCHEMBL4479032 0.78 ADRB3 (0.60) ADRB3ADRB1ADRB2GLA
SCHEMBL4462538 0.78 ADRB3 (0.60) ADRB3ADRB1ADRB2GLABACE1
SCHEMBL4468301 0.78 ADRB3 (0.59) ADRB3ADRB1ADRB2GLA
SCHEMBL4468296 0.78 ADRB3 (0.59) ADRB3ADRB1ADRB2GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993010074-A1 ARYLETHANOLAMINE DERIVATIVES AND THEIR USE AS BETA-3-ADRENOCEPTOR AGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-05-27 WO disclosed