SCHEMBL9547679

SCHEMBL9547679

Nc1nc(N)c2nc(CCc3ccnc(C(=O)O)c3)cnc2n1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 0.51
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA9 Q16790 1/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9315011 0.87 DHFR (0.48) DHFRCA1CA2
SCHEMBL24344752 0.81 DHFR (0.65) DHFRCA1CA2CA9
SCHEMBL24344201 0.75 DHFR (0.61) DHFRCA1CA2CA9
SCHEMBL9067320 0.74 DHFR (0.47) DHFRCA1CA2
SCHEMBL10582322 0.73 DHFR (0.59) DHFRCA1CA2CA9MEN1
SCHEMBL24344794 0.73 DHFR (0.58) DHFRCA1CA2CA9
SCHEMBL22679863 0.73 DHFR (0.66) DHFR
SCHEMBL3434673 0.70 DHFR (0.65) DHFRCA1CA2CA9
SCHEMBL30433658 0.70 DHFR (0.50) DHFR
SCHEMBL23996314 0.70 DHFR (0.69) DHFRCA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993022315-A1 HETEROAROYL-10-DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION SRI INTERNATIONAL (US) 1993-11-11 WO disclosed