SCHEMBL9557665

SCHEMBL9557665

N#CC(CBr)(CCc1cccc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.48
MIF P14174 2/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
GRM2 Q14416 1/20 0.41
GRM3 Q14832 1/20 0.41
IDO1 P14902 2/20 0.40
ATM Q13315 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9557571 0.90 CNR1 (0.44) TAAR1MIFMEN1KMT2AGRM2
SCHEMBL11825679 0.80 TAAR1 (0.56) TAAR1MIFMEN1KMT2AGRM2
SCHEMBL9556996 0.77 HSP90AA1 (0.43) TAAR1MIFKDM4ECYP1A2CYP3A4
SCHEMBL27709750 0.76 CCR1 (0.40) TAAR1ATMSIGMAR1
SCHEMBL9804762 0.74 CTSC (0.39) TAAR1MIFMEN1KMT2AGRIN1
Hydrochloric Acid SCHEMBL10925068 0.74 CYP2D6 (0.47) TAAR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL9557205 0.73 LTA4H (0.41) TAAR1MEN1KMT2AATMALDH1A1
SCHEMBL177514 0.72 TAAR1 (0.67) TAAR1MIFMEN1KMT2AIDO1
SCHEMBL30186510 0.72 TAAR1 (0.67) TAAR1MIFMEN1KMT2AIDO1
SCHEMBL8781661 0.72 TAAR1 (0.67) TAAR1MIFMEN1KMT2AGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0251775-B1 ALPHA-ARYL-ALPHA-PHENYLETHYL-1H-1,2,4-TRIAZOLE-1-PROPANENITRILES ROHM AND HAAS COMPANY (US) 1993-01-20 EP disclosed
US-5087635-A Funcicides ROHM AND HAAS COMPANY (US) 1992-02-11 US disclosed
EP-0251775-A2 Alpha-aryl-alpha-phenylethyl-1H-1,2,4-triazole-1-propanenitriles ROHM AND HAAS COMPANY (US) 1988-01-07 EP disclosed