SCHEMBL955786

SCHEMBL955786

CC(=O)ON1C(=O)C2(NC(=O)N(Cc3cc(Cl)ccc3F)C2=O)c2c1ccc(Cl)c2C(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 16/20 0.54
AKR1B1 P15121 1/20 0.40
UCHL3 P15374 2/20 0.37
UCHL1 P09936 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10025241 0.71 PTGDR2 (0.74) PTGDR2AKR1B1
SCHEMBL958668 0.70 PTGDR2 (1.00) PTGDR2AKR1B1
SCHEMBL954381 0.70 PTGDR2 (0.67) PTGDR2AKR1B1
SCHEMBL11959126 0.66 PTGDR2 (0.75) PTGDR2AKR1B1
SCHEMBL6127700 0.66 PTGDR2 (0.61) PTGDR2AKR1B1
SCHEMBL2483180 0.64 PTGDR2 (1.00) PTGDR2AKR1B1
SCHEMBL2486352 0.64 PTGDR2 (0.62) PTGDR2AKR1B1
SCHEMBL2484248 0.58 PTGDR2 (0.64) PTGDR2
SCHEMBL11959124 0.58 PTGDR2 (0.59) PTGDR2
SCHEMBL10025212 0.58 PTGDR2 (1.00) PTGDR2AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006936-A1 TRICYCLIC INDOLE-DERIVED SPIRO DERIVATIVES AS CRTH2 MODULATORS MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed