SCHEMBL9564273

SCHEMBL9564273

Cc1nc(O)c2c(C(C)c3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)c[nH]c2n1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHFR P00374 8/20 0.52
TYMS P04818 8/20 0.52
GART P22102 7/20 0.47
FOLR2 P14207 1/20 0.47
FOLR1 P15328 1/20 0.47
ATIC P31939 1/20 0.47
SHMT1 P34896 1/20 0.47
SLC19A1 P41440 1/20 0.47
FRK P42685 1/20 0.47
SLC46A1 Q96NT5 1/20 0.47
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564177 0.91 DHFR (0.52) DHFRTYMSGARTFOLR2FOLR1
SCHEMBL9564201 0.90 TYMS (0.51) DHFRTYMSGARTFOLR2FOLR1
SCHEMBL9564174 0.90 DHFR (0.60) DHFRTYMSGARTFOLR2FOLR1
SCHEMBL9564153 0.89 TYMS (0.49) DHFRTYMSGARTFOLR2FOLR1
SCHEMBL9564158 0.89 TYMS (0.51) DHFRTYMSGARTFOLR2FOLR1
SCHEMBL9564157 0.89 TYMS (0.49) DHFRTYMSGARTFOLR2FOLR1
SCHEMBL9564197 0.88 TYMS (0.50) DHFRTYMSGARTFOLR2FOLR1
SCHEMBL9564176 0.88 TYMS (0.52) DHFRTYMSGARTFOLR2FOLR1
SCHEMBL9564147 0.88 TYMS (0.50) DHFRTYMSGARTFOLR2FOLR1
SCHEMBL9564173 0.88 TYMS (0.49) DHFRTYMSGARTFOLR2FOLR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549291-A1 Thymidylate synthase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-30 EP disclosed