SCHEMBL9564539

SCHEMBL9564539

NCCCCc1ccc2occc2c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 4/20 0.46
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
MAOA P21397 1/20 0.41
TLR8 Q9NR97 4/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
DYRK1A Q13627 3/20 0.40
CDK9 P50750 1/20 0.40
CYP2A6 P11509 2/20 0.40
HRH1 P35367 2/20 0.38
BCDIN3D Q7Z5W3 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4451104 0.87 HTR1B (0.50) HTR1BCYP1A2CYP2D6DYRK1ACDK9
SCHEMBL25742668 0.84 HTR1B (0.47) HTR1BCYP1A2CYP2D6CYP2C19CHRM2
SCHEMBL7472414 0.83 HTR1B (0.51) HTR1BTLR8CHRM2CHRM1CHRM3
SCHEMBL826348 0.83 HTR1B (0.46) HTR1BMAOACHRM2CHRM1CHRM3
SCHEMBL28493440 0.81 HTR1B (0.50) HTR1BTLR8CHRM2CHRM1CHRM3
SCHEMBL1603347 0.81 HTR1B (0.53) HTR1BCHRM2CHRM1CHRM3CYP2A6
SCHEMBL28326818 0.81 HTR1B (0.47) HTR1BCHRM2CHRM1CHRM3DYRK1A
SCHEMBL31164857 0.80 CA2 (0.55) HTR1BDYRK1ACDK9CYP2A6BCDIN3D
SCHEMBL111709 0.80 CA2 (0.55) HTR1BDYRK1ACDK9CYP2A6BCDIN3D
Ammonia Solution, Strong SCHEMBL9564542 0.79 HTR1B (0.51) HTR1BCHRM2CHRM1CHRM3CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533265-A1 Process of making substituted azetidinones MERCK & CO. INC. (US) 1993-03-24 EP disclosed
US-5149838-A Intermediates for substituted azetidinones useful as anti-inflammatory and antidegenerative agents MERCK & CO., INC. (US) 1992-09-22 US disclosed