SCHEMBL9564944

SCHEMBL9564944

COc1ccc(CCN2CCC(N(C)c3nc4cncnc4n3Cc3ccc(F)cc3)CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 8/20 0.50
CYP3A4 P08684 7/20 0.50
CYP2C19 P33261 6/20 0.50
USP2 O75604 6/20 0.50
LMNA P02545 4/20 0.50
HRH1 P35367 3/20 0.50
CYP2D6 P10635 3/20 0.50
TACR2 P21452 2/20 0.50
TACR1 P25103 2/20 0.50
EED O75530 2/20 0.50
KCNH2 Q12809 2/20 0.50
SSTR5 P35346 2/20 0.50
HTR1A P08908 2/20 0.50
SLC6A4 P31645 2/20 0.50
MEN1 O00255 1/20 0.50
MLNR O43193 1/20 0.50
CACNA1F O60840 1/20 0.50
ABCB11 O95342 1/20 0.50
EGFR P00533 1/20 0.50
HLA-A P04439 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564844 0.78 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C19USP2LMNA
Fumaric Acid SCHEMBL9876528 0.77 HRH1 (0.49) CYP1A2CYP3A4CYP2C19USP2LMNA
Hydrochloric Acid SCHEMBL11470684 0.75 SSTR5 (0.65) CYP1A2CYP3A4CYP2C19USP2LMNA
SCHEMBL9564763 0.71 CYP1A2 (0.54) CYP1A2CYP3A4CYP2C19USP2LMNA
SCHEMBL9564878 0.71 HRH1 (0.49) CYP1A2CYP3A4CYP2C19USP2LMNA
SCHEMBL10547773 0.71 HTR1A (0.56) CYP1A2CYP3A4CYP2C19USP2LMNA
SCHEMBL1151577 0.70 KCNH2 (0.80) CYP1A2CYP3A4CYP2C19USP2LMNA
SCHEMBL9565053 0.69 KCNH2 (0.57) CYP1A2CYP3A4CYP2C19USP2LMNA
SCHEMBL11482399 0.68 HRH1 (0.58) CYP1A2CYP3A4CYP2C19USP2LMNA
SCHEMBL10428778 0.68 KCNH2 (0.80) CYP1A2CYP3A4CYP2C19USP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed