SCHEMBL9564960

SCHEMBL9564960

c1csc(Cn2c(NC3CCNCC3)nc3cncnc32)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 19/20 0.43
CYP3A4 P08684 19/20 0.43
ALDH1A1 P00352 18/20 0.43
CYP2D6 P10635 8/20 0.43
HPGD P15428 5/20 0.43
HSD17B10 Q99714 11/20 0.43
NR4A2 P43354 1/20 0.42
KCNH2 Q12809 1/20 0.42
CYP2C9 P11712 14/20 0.42
CASP1 P29466 13/20 0.42
CASP7 P55210 12/20 0.42
CYP2C19 P33261 11/20 0.42
USP2 O75604 10/20 0.42
HIF1A Q16665 8/20 0.42
TP53 P04637 7/20 0.42
LMNA P02545 6/20 0.42
CLK4 Q9HAZ1 5/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
BLM P54132 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10428775 0.86 NR4A2 (0.46) CYP1A2CYP3A4ALDH1A1CYP2D6HPGD
SCHEMBL9564905 0.84 CYP1A2 (0.37) CYP1A2CYP3A4ALDH1A1CYP2D6HPGD
Bromide SCHEMBL9564796 0.82 NR4A2 (0.54) CYP1A2CYP3A4ALDH1A1CYP2D6HPGD
SCHEMBL9564789 0.82 NR4A2 (0.42) CYP1A2CYP3A4ALDH1A1CYP2D6HPGD
Water SCHEMBL9564806 0.81 NR4A2 (0.42) CYP1A2CYP3A4ALDH1A1CYP2D6HPGD
Water SCHEMBL9564807 0.81 NR4A2 (0.42) CYP1A2CYP3A4ALDH1A1CYP2D6HPGD
SCHEMBL9564782 0.81 KCNH2 (0.45) CYP1A2CYP3A4ALDH1A1CYP2D6HSD17B10
SCHEMBL9564849 0.80 SMN1; SMN2 (0.50) ALDH1A1CYP2D6HPGDHSD17B10LMNA
SCHEMBL9698816 0.80 KCNH2 (0.65) HPGDHSD17B10NR4A2KCNH2ALOX15
SCHEMBL9631535 0.80 MAPT (0.42) CYP1A2CYP3A4ALDH1A1CYP2D6HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed