SCHEMBL9565491

SCHEMBL9565491

O[C@H]1C[C@](F)(COCc2ccccc2)C1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
TACR1 P25103 2/20 0.42
CA1 P00915 3/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
EPHX2 P34913 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9565489 1.00 TSHR (0.45) TSHRTACR1CA1CA2CA7
SCHEMBL28306256 0.80 TSHR (0.54) TSHRTACR1CA1CA2CA7
SCHEMBL2221074 0.76 TSHR (0.48) TSHRTACR1CA1CA2CA7
SCHEMBL763893 0.76 TSHR (0.48) TSHRTACR1CA1CA2CA7
SCHEMBL1857389 0.76 TSHR (0.48) TSHRTACR1CA1CA2CA7
SCHEMBL1857390 0.76 TSHR (0.48) TSHRTACR1CA1CA2CA7
SCHEMBL599239 0.75 TSHR (0.47) TSHRTACR1
SCHEMBL26124613 0.75 TSHR (0.47) TSHRTACR1CA1CA2CA7
SCHEMBL9565492 0.74 TSHR (0.39) TSHRTACR1EPHX2
SCHEMBL9565495 0.74 TSHR (0.39) TSHRTACR1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0554025-A2 Fluorinated cyclobutyl purines and pyrimidines E.R. SQUIBB & SONS, INC. (US) 1993-08-04 EP disclosed