SCHEMBL9565545

SCHEMBL9565545

c1nc2cnc(C3CCC3)nc2[nH]1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CDK5 Q00535 1/20 0.34
ALOX5AP P20292 2/20 0.34
FEN1 P39748 2/20 0.34
PAK1 Q13153 2/20 0.32
LMNA P02545 1/20 0.30
HTT P42858 1/20 0.30
AURKA O14965 1/20 0.30
JAK1 P23458 1/20 0.30
TYK2 P29597 1/20 0.30
KDR P35968 1/20 0.30
FLT3 P36888 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30
CHRM3 P20309 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946172 0.97 PAK1 (0.35) CCNE1CDK2CDK5ALOX5APFEN1
SCHEMBL10600434 0.95 PAK1 (0.37) PAK1LMNAHTTAURKAJAK1
Hydrochloric Acid SCHEMBL6821627 0.95 PAK1 (0.34) CCNE1CDK2CDK5ALOX5APFEN1
SCHEMBL4373719 0.81 HRH3 (0.36)
SCHEMBL9854783 0.77 MAPK8 (0.30)
SCHEMBL4156180 0.76 MAPK8 (0.35) PAK1AURKAKDM4EALDH1A1
SCHEMBL2953146 0.76
SCHEMBL28057563 0.75 MAPK8 (0.39) PAK1
SCHEMBL8710206 0.75
SCHEMBL1551868 0.73 PAK1 (0.56) PAK1LMNAHTTFLT3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2377865-B1 CYCLOBUTYL PURINE DERIVATIVE, ANGIOGENESIS PROMOTING AGENT, LUMENIZATION PROMOTING AGENT, NEUROCYTE GROWTH PROMOTING AGENT, AND DRUG UNIV KAGAWA NAT UNIV CORP (JP) 2014-12-17 EP claimed
EP-0554025-A2 Fluorinated cyclobutyl purines and pyrimidines E.R. SQUIBB & SONS, INC. (US) 1993-08-04 EP disclosed