SCHEMBL9565771

SCHEMBL9565771

COc1cccc(C(O)C2CC(=O)CCN2C(=O)c2cc(C)cc(C)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 1/20 0.42
GRIN2C Q14957 2/20 0.38
MTNR1B P49286 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TACR1 P25103 2/20 0.36
ABCB1 P08183 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD11B1 P28845 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8927584 1.00 HSD17B2 (0.42) HSD17B2GRIN2CMTNR1BL3MBTL1TACR1
SCHEMBL8923597 1.00 HSD17B2 (0.42) HSD17B2GRIN2CMTNR1BL3MBTL1TACR1
SCHEMBL8926073 0.90 GRIN2C (0.40) HSD17B2GRIN2CTACR1MEN1KMT2A
SCHEMBL8925866 0.90 GRIN2C (0.40) HSD17B2GRIN2CTACR1MEN1KMT2A
SCHEMBL9204527 0.86 TACR1 (0.41) HSD17B2MTNR1BTACR1
SCHEMBL8939874 0.86 TACR1 (0.41) HSD17B2MTNR1BTACR1
SCHEMBL8926027 0.81 HSD17B2 (0.40) HSD17B2TACR1OPRK1
SCHEMBL8925651 0.81 HSD17B2 (0.40) HSD17B2TACR1OPRK1
SCHEMBL8924315 0.81 HSD17B2 (0.36) HSD17B2TACR1
SCHEMBL8925754 0.81 HSD17B2 (0.36) HSD17B2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0532456-A1 1-Acylpiperidine derivatives and their use as substance P antagonists CIBA-GEIGY AG (CH) 1993-03-17 EP claimed