SCHEMBL9566934

SCHEMBL9566934

COC(=O)C(=O)c1c(OCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cccc1C1CCCCN1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.40
MAOB P27338 2/20 0.40
HIF1A Q16665 1/20 0.39
TP53 P04637 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
TSHR P16473 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
THPO P40225 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GMNN O75496 1/20 0.38
LMNA P02545 1/20 0.38
PMP22 Q01453 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2987773 0.70 TACR1 (0.52) TACR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL9025417 0.70 TACR1 (0.52) TACR1TP53CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9024656 0.70 MEN1 (0.43) TACR1MAOBTP53CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL8546078 0.70 MEN1 (0.53) TACR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL8867313 0.67 TACR1 (0.53) TACR1TP53CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9025813 0.67 HTR6 (0.45) TACR1MAOBCYP1A2CYP2D6TSHR
Hydrochloric Acid SCHEMBL8116324 0.67 MEN1 (0.54) TACR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL31136940 0.66 MEN1 (0.60) MEN1KMT2A
Acetic Acid SCHEMBL27852935 0.64 PTGDR2 (0.39) TACR1MEN1KMT2ALMNAPMP22
Acetic Acid SCHEMBL27853031 0.63 CYP11B1 (0.41) TSHRMEN1KMT2ALMNAPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528495-A1 Azacyclic compounds, processes for their preparation and pharmaceutical compositions containing them MERCK SHARP & DOHME LTD. (GB) 1993-02-24 EP disclosed