SCHEMBL9569109

SCHEMBL9569109

C#Cc1cccc(Cc2ccccc2)c1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.40
CALM1 P0DP23 1/20 0.39
BCL2 P10415 1/20 0.38
BCL2L1 Q07817 1/20 0.38
CYP3A4 P08684 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
ALOX5 P09917 1/20 0.34
HPGD P15428 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
DAO P14920 1/20 0.33
PDE2A O00408 1/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2870972 0.84 CALM1 (0.46) HTR2ACALM1BCL2BCL2L1CYP3A4
SCHEMBL7735333 0.80 CALM1 (0.55) HTR2ACALM1BCL2BCL2L1CYP3A4
SCHEMBL10360527 0.76 HTR2A (0.54) HTR2ACALM1BCL2BCL2L1CYP3A4
SCHEMBL1046166 0.73 CALM1 (0.58) HTR2ACALM1BCL2BCL2L1CYP3A4
SCHEMBL29532678 0.72 IDH1 (0.47) HTR2ACALM1BCL2BCL2L1CYP3A4
SCHEMBL9719201 0.72 IDH1 (0.47) HTR2ACALM1BCL2BCL2L1CYP3A4
SCHEMBL146769 0.72 IDH1 (0.47) HTR2ACALM1BCL2BCL2L1CYP3A4
SCHEMBL1838403 0.71 BCL2 (0.57) HTR2ACALM1BCL2BCL2L1CYP3A4
SCHEMBL7033288 0.71 HPGD (0.49) HTR2ACALM1BCL2BCL2L1CYP3A4
SCHEMBL9419606 0.71 CALM1 (0.44) HTR2ACALM1BCL2BCL2L1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0565450-A1 Use of peptide derivatives for the manufacture of medicaments inhibiting endopeptidases 24.15 and 24.16 COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 1993-10-13 EP disclosed