SCHEMBL9569155

SCHEMBL9569155

C=CC(N)COCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.54
CA1 P00915 4/20 0.51
CA2 P00918 2/20 0.51
CA7 P43166 2/20 0.51
CA9 Q16790 2/20 0.51
TSHR P16473 1/20 0.50
SLC1A1 P43005 1/20 0.47
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.43
IDO1 P14902 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4410718 0.98 TACR1 (0.53) TACR1CA1CA2CA7CA9
SCHEMBL14401030 0.81 TACR1 (0.54) TACR1CA1CA2CA7CA9
SCHEMBL13354771 0.81 TACR1 (0.54) TACR1CA1CA2CA7CA9
SCHEMBL13267636 0.81 TACR1 (0.58) TACR1CA1CA2CA7CA9
SCHEMBL2997911 0.81 TACR1 (0.58) TACR1CA1CA2CA7CA9
SCHEMBL2997913 0.81 TACR1 (0.58) TACR1CA1CA2CA7CA9
Hydrochloric Acid SCHEMBL16993593 0.80 TACR1 (0.53) TACR1CA1CA2CA7CA9
SCHEMBL17688799 0.79 TACR1 (0.51) TACR1CA1CA2CA7CA9
SCHEMBL2989933 0.79 TACR1 (0.51) TACR1CA1CA2CA7CA9
SCHEMBL22013212 0.78 TACR1 (0.63) TACR1CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1079745-A New 9-fluoro-7-oxo-7H-pyrido [1,2,3-d, e] [1,4] benzoxazine-6-carboxylic acids and ester thereof BAYER AG (DE) 1993-12-22 CN disclosed
EP-0563734-A1 9-fluoro-7-oxo-7H-pyrido(1,2,3-de)(1,4)benzoxazine carboxylic acids and esters and their use as antiviral agents BAYER AG (DE) 1993-10-06 EP disclosed