SCHEMBL9569321

SCHEMBL9569321

CN(C)c1nc(N)nc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)C1(F)F

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.49
CYP2C19 P33261 1/20 0.48
SLC29A1 Q99808 8/20 0.47
PDE4D Q08499 1/20 0.47
PDE3A Q14432 1/20 0.47
ADORA3 P0DMS8 2/20 0.45
ADORA1 P30542 2/20 0.45
ADA P00813 1/20 0.44
PGK1 P00558 1/20 0.42
PGK2 P07205 1/20 0.42
LMNA P02545 1/20 0.41
NT5E P21589 1/20 0.41
HIF1A Q16665 1/20 0.41
ADORA2B P29275 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18061793 0.91 ADORA2A (0.51) ADORA2ACYP2C19SLC29A1ADORA3ADORA1
SCHEMBL18041236 0.91 ADORA2A (0.51) ADORA2ACYP2C19SLC29A1ADORA3ADORA1
SCHEMBL22224923 0.88 ADORA2A (0.65) ADORA2ACYP2C19SLC29A1ADORA3ADORA1
SCHEMBL21136193 0.88 ADORA2A (0.65) ADORA2ACYP2C19SLC29A1ADORA3ADORA1
SCHEMBL2503256 0.88 ADORA2A (0.65) ADORA2ACYP2C19SLC29A1ADORA3ADORA1
SCHEMBL23761057 0.88 ADORA2A (0.65) ADORA2ACYP2C19SLC29A1ADORA3ADORA1
SCHEMBL21136198 0.87 ADORA2A (0.46) ADORA2ACYP2C19SLC29A1ADORA3ADORA1
SCHEMBL21137196 0.87 ADORA2A (0.46) ADORA2ACYP2C19SLC29A1ADORA3ADORA1
SCHEMBL18061771 0.87 ADORA2A (0.46) ADORA2ACYP2C19SLC29A1ADORA3ADORA1
SCHEMBL18061805 0.87 ADORA2A (0.46) ADORA2ACYP2C19SLC29A1ADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0576227-A2 2'-Deoxy-2',2'-difluoro(2,6,8-substituted) purine nucleosides having anti-viral and anti-cancer activity and intermediates ELI LILLY AND COMPANY (US) 1993-12-29 EP claimed
EP-0576227-A2 2'-Deoxy-2',2'-difluoro(2,6,8-substituted) purine nucleosides having anti-viral and anti-cancer activity and intermediates ELI LILLY AND COMPANY (US) 1993-12-29 EP disclosed