SCHEMBL9570448

SCHEMBL9570448

O=C(O)Nn1nc(Cc2ccccc2)c2ccccc2c1=O

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.62
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
GLA P06280 1/20 0.48
ALDH1A1 P00352 3/20 0.43
ENPP1 P22413 1/20 0.43
PARP1 P09874 1/20 0.43
AR P10275 1/20 0.43
CMA1 P23946 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ALOX15 P16050 1/20 0.43
POLB P06746 1/20 0.42
PKM P14618 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7892953 0.84 TSHR (0.54) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1788819 0.81 TSHR (0.51) TSHRALDH1A1MEN1KMT2A
SCHEMBL30796387 0.81 TSHR (0.51) TSHRALDH1A1MEN1KMT2A
SCHEMBL30795814 0.81 TSHR (0.50) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL30796305 0.81 TSHR (0.50) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1786762 0.81 TSHR (0.50) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1791416 0.81 TSHR (0.50) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1790428 0.78 ADRA1A (0.51) TSHRALDH1A1MEN1KMT2A
SCHEMBL30795062 0.78 ADRA1A (0.51) TSHRALDH1A1MEN1KMT2A
SCHEMBL1788569 0.77 TSHR (0.46) TSHRCYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564805-A1 (4-benzylphthalazin-1(2H)-on-2-yl)aminocarboxylic acids having antiallergic/antihistaminic activity and process for their production ASTA Medica Aktiengesellschaft (DE) 1993-10-13 EP disclosed