SCHEMBL9573545

SCHEMBL9573545

O=C1Nc2ccccc2C(c2ccccc2)=NC1N(Cc1ccccc1)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.54
ALDH1A1 P00352 1/20 0.54
KMT2A Q03164 1/20 0.54
CCKBR P32239 15/20 0.53
CCKAR P32238 11/20 0.53
HDAC1 Q13547 1/20 0.51
BACE1 P56817 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16777948 0.84 NOTCH1 (0.49) MEN1ALDH1A1KMT2ACCKBRCCKAR
SCHEMBL16777944 0.84 CCKBR (0.40) MEN1ALDH1A1KMT2ACCKBRCCKAR
SCHEMBL16777947 0.84 NOTCH1 (0.49) MEN1ALDH1A1KMT2ACCKBRCCKAR
SCHEMBL16777930 0.83 MEN1 (0.44) MEN1ALDH1A1KMT2ACCKBRCCKAR
SCHEMBL16777950 0.82 NOTCH1 (0.51) MEN1ALDH1A1KMT2ACCKBRCCKAR
SCHEMBL24612375 0.78 CCKBR (0.51) MEN1ALDH1A1KMT2ACCKBRCCKAR
SCHEMBL8741334 0.78 CCKBR (0.58) MEN1ALDH1A1KMT2ACCKBRCCKAR
SCHEMBL15608190 0.77 NOTCH1 (0.51) CCKBRCCKAR
SCHEMBL15608191 0.77 NOTCH1 (0.51) CCKBRCCKAR
SCHEMBL24611851 0.77 CCKBR (0.53) MEN1ALDH1A1KMT2ACCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993008175-A1 BENZODIAZEPINE DERIVATIVES AS ANTAGONISTS OF GASTRIN AND/OR CHOLECYSTOKININ GLAXO GROUP LIMITED (GB) 1993-04-29 WO disclosed
EP-0538945-A1 Benzodiazepine derivatives, and their use as antagonists of gastrin and/or cholecystokinin GLAXO GROUP LIMITED (GB) 1993-04-28 EP disclosed