SCHEMBL9586019

SCHEMBL9586019

NCCNC(=O)c1ncsc1-c1cc(F)cc(F)c1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.78
CYP3A4 P08684 1/20 0.78
THPO P40225 1/20 0.78
PMP22 Q01453 2/20 0.76
LMNA P02545 1/20 0.76
CHEK1 O14757 3/20 0.36
CHEK2 O96017 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MAOB P27338 2/20 0.36
TDO2 P48775 1/20 0.35
ADORA2A P29274 1/20 0.35
HSD17B13 Q7Z5P4 1/20 0.34
FPR2 P25090 1/20 0.34
TERT O14746 2/20 0.33
HCRTR2 O43614 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
AKT1 P31749 1/20 0.33
SPHK2 Q9NRA0 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9585626 0.99 PMP22 (0.78) CYP1A2CYP3A4THPOPMP22LMNA
SCHEMBL6866198 0.88 CYP1A2 (1.00) CYP1A2CYP3A4THPOPMP22LMNA
SCHEMBL9586566 0.87 CYP1A2 (0.60) CYP1A2CYP3A4THPOPMP22LMNA
SCHEMBL9585836 0.87 CYP1A2 (0.74) CYP1A2CYP3A4THPOPMP22LMNA
Hydrochloric Acid SCHEMBL1665880 0.87 LMNA (1.00) CYP1A2CYP3A4THPOPMP22LMNA
Hydrochloric Acid SCHEMBL9585703 0.86 PMP22 (0.74) CYP1A2CYP3A4THPOPMP22LMNA
SCHEMBL9586484 0.84 CYP1A2 (0.63) CYP1A2CYP3A4THPOPMP22LMNA
Hydrochloric Acid SCHEMBL9586454 0.84 PMP22 (0.75) CYP1A2CYP3A4THPOPMP22LMNA
Hydrochloric Acid SCHEMBL9586753 0.83 PMP22 (0.64) CYP1A2CYP3A4THPOPMP22LMNA
SCHEMBL9586621 0.81 CYP1A2 (0.73) CYP1A2CYP3A4THPOPMP22LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011849-A Monoamine oxidase inhibitors HOFFMANN-LA ROCHE INC. (US) 1991-04-30 US claimed
US-5204482-A Ethylenediamine monoamide heteroaryl derivatives HOFFMAN-LAROCHE INC. (US) 1993-04-20 US disclosed
US-5011849-A Monoamine oxidase inhibitors HOFFMANN-LA ROCHE INC. (US) 1991-04-30 US disclosed
EP-0352581-A2 Ethylene diaminmonoamide derivatives F. HOFFMANN-LA ROCHE AG (CH) 1990-01-31 EP disclosed