SCHEMBL9586755

SCHEMBL9586755

CNc1ccc(N)c(C#N)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43
KDM4E B2RXH2 3/20 0.40
MAPT P10636 2/20 0.40
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 5/20 0.37
USP2 O75604 1/20 0.35
CHUK O15111 1/20 0.33
IDO1 P14902 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12272254 0.84 KDM4E (0.40) CYP1A2CYP3A4TSHRMAPK1ADRB2
SCHEMBL28643560 0.83 KDM4E (0.46) CYP1A2CYP3A4TSHRMAPK1ADRB2
SCHEMBL14046649 0.81 ALDH1A1 (0.46) KDM4EMAPTGAAMEN1LMNA
SCHEMBL9587134 0.79 CYP1A2 (0.43) CYP1A2CYP3A4TSHRMAPK1ADRB2
SCHEMBL21966924 0.78 TSHR (0.45) TSHRKDM4EMAPTHTTSMN1; SMN2
SCHEMBL3173181 0.78 GRM4 (0.48) MAPTLMNAALDH1A1ABCG2
SCHEMBL6815182 0.77 ALDH1A1 (0.63) CYP3A4TSHRKDM4EMAPTMEN1
SCHEMBL8343255 0.76 SLC22A12 (0.50) MAPTALDH1A1IDO1
SCHEMBL12117937 0.73 ABCG2 (0.46) TSHRMAPTHTTALDH1A1ABCG2
SCHEMBL13548437 0.73 TDP1 (0.46) CYP3A4TSHRMEN1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013079-A1 ANTIFOLATE QUINAZOLINES AGOURON PHARMACEUTICALS, INC. (US) 1993-07-08 WO disclosed