SCHEMBL9587719

SCHEMBL9587719

Cc1[nH]c(=O)c(-c2nnn[nH]2)cc1Sc1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 4/20 0.35
BRD4 O60885 3/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
PNP P00491 1/20 0.33
KDM4E B2RXH2 2/20 0.32
NSD2 O96028 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
POLB P06746 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
DHFR P00374 1/20 0.32
ALDH1A1 P00352 2/20 0.32
GAA P10253 2/20 0.32
ADORA2A P29274 1/20 0.32
GALR3 O60755 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9590686 0.88 TYMS (0.42) TYMSDHFRMAOAMAOB
SCHEMBL9378837 0.88 TYMS (0.37) TYMSMAPK1DHFRGAAMAOA
SCHEMBL9377783 0.87 TYMS (0.42) TYMSKDM4EDHFRALDH1A1HPGD
SCHEMBL9375105 0.84 PTPN11 (0.34) TYMSPOLBL3MBTL1DHFR
SCHEMBL9589264 0.84 PNP (0.32) TYMSPNPKDM4ENSD2MAPT
SCHEMBL9588530 0.83 TYMS (0.41) TYMSL3MBTL1DHFRALDH1A1
SCHEMBL9374084 0.80 KDR (0.35) KDM4EMAPTMAPK1POLBALDH1A1
SCHEMBL9374095 0.80 KDR (0.35) KDM4EMAPTMAPK1POLBALDH1A1
SCHEMBL9587889 0.78 MAPK8 (0.36) TYMSMAOB
SCHEMBL9590145 0.75 TYMS (0.37) TYMSPDE3BPDE3ADHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993007137-A1 PYRIDINOL DERIVATIVES AS MEDICAMENTS SMITHKLINE BEECHAM PLC (GB) 1993-04-15 WO claimed
WO-1993007137-A1 PYRIDINOL DERIVATIVES AS MEDICAMENTS SMITHKLINE BEECHAM PLC (GB) 1993-04-15 WO disclosed