SCHEMBL9588404

SCHEMBL9588404

[CH2][C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.61
CTSS P25774 5/20 0.59
CTSK P43235 4/20 0.59
CTSB P07858 2/20 0.59
CTSL P07711 1/20 0.59
ACE P12821 1/20 0.56
KLK5 Q9Y337 2/20 0.52
PPARA Q07869 2/20 0.51
PPARG P37231 1/20 0.51
AKT1 P31749 1/20 0.51
APP P05067 2/20 0.50
ALDH1A1 P00352 2/20 0.50
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.49
PKM P14618 1/20 0.49
HPGD P15428 1/20 0.49
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.49
XBP1 P17861 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7349815 1.00 ATM (0.61) ATMCTSSCTSKCTSBCTSL
SCHEMBL27759656 0.87 CTSS (0.58) ATMCTSSCTSKCTSBCTSL
SCHEMBL20397779 0.85 PPARG (0.51) ATMCTSSCTSKCTSBCTSL
SCHEMBL7425280 0.84 KLK5 (0.61) ATMCTSSCTSKCTSBCTSL
SCHEMBL20397698 0.84 PPARG (0.52) ATMCTSSCTSKCTSBCTSL
SCHEMBL6832510 0.84 KLK5 (0.61) ATMCTSSCTSKCTSBCTSL
SCHEMBL7939304 0.83 ATM (0.63) ATMCTSSCTSKCTSBCTSL
SCHEMBL3676166 0.83 NPC1 (0.63) ATMCTSSCTSKCTSBCTSL
SCHEMBL12203694 0.83 NPC1 (0.63) ATMCTSSCTSKCTSBCTSL
SCHEMBL3676162 0.83 NPC1 (0.63) ATMCTSSCTSKCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117486762-A Novel compound and use method and application thereof 中国医学科学院医药生物技术研究所 2024-02-02 CN disclosed
EP-2809646-A1 METHODS AND INTERMEDIATES FOR PREPARING PHARMACEUTICAL AGENTS Gilead Sciences, Inc. (US) 2014-12-10 EP disclosed
WO-2013116715-A1 METHODS AND INTERMEDIATES FOR PREPARING PHARMACEUTICAL AGENTS GILEAD SCIENCES, INC. (US) 2013-08-08 WO disclosed
US-5190974-A Analgesics ROUSSEL UCLAF (FR) 1993-03-02 US disclosed
CN-1049165-A The cycloalkyl that N-replaces and the tryptophane-phenylalanine of multi-ring alkyl alpha-substitution-and phenylethylamine derivative WARNER LAMBERT CO (US) 1991-02-13 CN disclosed