SCHEMBL9595376

SCHEMBL9595376

CC(C)(C)OC(=O)N1CC(O[Si](C)(C)C(C)(C)C)C[C@H]1C=O

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
ALDH1A1 P00352 2/20 0.34
PPM1D O15297 1/20 0.33
TSHR P16473 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PARP1 P09874 1/20 0.32
RECQL P46063 1/20 0.32
USP2 O75604 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15632355 1.00 NR1H2 (0.36) NR1H2CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL27274652 1.00 NR1H2 (0.36) NR1H2CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL31234239 1.00 NR1H2 (0.36) NR1H2CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL144330 1.00 NR1H2 (0.36) NR1H2CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL141264 1.00 NR1H2 (0.36) NR1H2CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL573307 1.00 NR1H2 (0.36) NR1H2CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL15632374 1.00 NR1H2 (0.36) NR1H2CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL1882303 1.00 NR1H2 (0.36) NR1H2CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL24540367 0.91 ALDH1A1 (0.36) CHRM2CHRM1CHRM3ALDH1A1TSHR
SCHEMBL23555453 0.91 ALDH1A1 (0.36) CHRM2CHRM1CHRM3ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022187206-A1 DUAL-TARGET MU OPIOID AND DOPAMINE D3 RECEPTORS LIGANDS; PREPARATION AND USE THEREOF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2022-09-09 WO disclosed
WO-1993011128-A1 AMINOALKYLPYRROLIDINYLTHIOCARBAPENEM DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-06-10 WO disclosed
WO-1993001174-A1 THIAZOLIDINE DERIVATIVES AND THEIR USE AS ANTI-VIRAL COMPOUNDS GLAXO GROUP LIMITED (GB) 1993-01-21 WO disclosed