SCHEMBL9598677

SCHEMBL9598677

O=c1nc2nc[nH]n2c2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 18/20 0.48
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7740293 0.71 HSD17B10 (0.43) KDM4ENPC1ALDH1A1TP53HPGD
SCHEMBL12883857 0.67 PARP1 (0.51) KDM4EALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL30773025 0.67 KDM4E (0.45) KDM4ENPC1ALDH1A1TP53HPGD
SCHEMBL203256 0.65 KDM5B (0.43) KDM5BKDM4ESMN1; SMN2
SCHEMBL7126019 0.64 KDM5B (0.44) KDM5BKDM4E
SCHEMBL7665757 0.64 KDM5B (0.44) KDM5B
SCHEMBL11447666 0.61 MAPK1 (0.59) KDM4EALDH1A1SMN1; SMN2HSD17B10
SCHEMBL17229160 0.61 KDM4E (0.53) KDM4ENPC1ALDH1A1TP53HPGD
SCHEMBL11779144 0.60 KDM4E (0.39) KDM4ENPC1ALDH1A1TP53HPGD
SCHEMBL20704529 0.60 HPGD (0.49) KDM4ENPC1ALDH1A1TP53HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993012113-A1 3-SUBSTITUTED IMIDAZO (1,5-a) AND IMIDAZO (1,5-a)-TRIAZOLO (1,5-c) QUINOXALINES AND QUINAZOLINES WITH CNS ACTIVITY THE UPJOHN COMPANY (US) 1993-06-24 WO disclosed