SCHEMBL9600313

SCHEMBL9600313

COC(=O)O[C@@H]1C=C[C@H](OC(C)=O)C1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.40
CA9 Q16790 4/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
ALDH1A1 P00352 1/20 0.35
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
TSHR P16473 2/20 0.32
ALOX5 P09917 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
HSD17B10 Q99714 1/20 0.30
KMT2A Q03164 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL254386 0.87 CA12 (0.42) CA12CA9CA1CA2CHRM2
SCHEMBL2290500 0.87 CA12 (0.42) CA12CA9CA1CA2CHRM2
SCHEMBL11746006 0.87 CA12 (0.42) CA12CA9CA1CA2CHRM2
SCHEMBL11548379 0.87 CA12 (0.42) CA12CA9CA1CA2CHRM2
SCHEMBL11548381 0.87 CA12 (0.42) CA12CA9CA1CA2CHRM2
SCHEMBL19464089 0.83 CA12 (0.38) CA12CA9CA1CA2ALDH1A1
SCHEMBL15750146 0.83 SLC6A4 (0.33)
SCHEMBL11835919 0.80 CA12 (0.40) CA12CA9CA1CA2TSHR
SCHEMBL9599191 0.80
SCHEMBL11835924 0.80 CA12 (0.40) CA12CA9CA1CA2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0489876-A1 SYNTHESIS OF CYCLOPENTENE DERIVATIVES GLAXO INC. (US) 1992-06-17 EP claimed
WO-1991015447-A1 SYNTHESIS OF CYCLOPENTENE DERIVATIVES GLAXO INC. (US) 1991-10-17 WO claimed
US-5241069-A Carbonate intermediates for the synthesis of purine substituted cyclopentene derivatives GLAXO INC. (US) 1993-08-31 US disclosed
US-5126452-A SYNTHESIS OF PURINE SUBSTITUTED CYCLOPENTENE DERIVATIVES GLAXO INC. (US) 1992-06-30 US disclosed
EP-0489876-A1 SYNTHESIS OF CYCLOPENTENE DERIVATIVES GLAXO INC. (US) 1992-06-17 EP disclosed
WO-1991015447-A1 SYNTHESIS OF CYCLOPENTENE DERIVATIVES GLAXO INC. (US) 1991-10-17 WO disclosed
US-5057630-A SYNTHESIS OF CYCLOPENTENE DERIVATIVES GLAXO INC. (US) 1991-10-15 US disclosed