SCHEMBL9601290

SCHEMBL9601290

CC(C[O])c1csc(N)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.42
NOS1 P29475 1/20 0.42
BACE1 P56817 1/20 0.38
HSD17B10 Q99714 2/20 0.38
GABRA5 P31644 1/20 0.38
GABRB2 P47870 1/20 0.38
ALDH1A1 P00352 6/20 0.37
NPC1 O15118 5/20 0.37
MAPT P10636 4/20 0.37
RAB9A P51151 4/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
GFER P55789 1/20 0.35
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
LTA4H P09960 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ADRB3 P13945 2/20 0.33
ATM Q13315 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10988006 0.82 SMN1; SMN2 (0.43) SMN1; SMN2NOS1BACE1HSD17B10GABRA5
SCHEMBL9601297 0.81 SMN1; SMN2 (0.42) SMN1; SMN2NOS1BACE1HSD17B10GABRA5
SCHEMBL12877376 0.79 NOS1 (0.41) SMN1; SMN2NOS1BACE1HSD17B10GABRA5
SCHEMBL190635 0.77
Bromide SCHEMBL5908220 0.75 SMN1; SMN2 (0.48) SMN1; SMN2NOS1BACE1HSD17B10ALDH1A1
SCHEMBL27677871 0.74 SMN1; SMN2 (0.43) SMN1; SMN2NOS1BACE1HSD17B10GABRA5
SCHEMBL14433411 0.74 BACE1 (0.59) SMN1; SMN2NOS1BACE1HSD17B10ALDH1A1
SCHEMBL14433410 0.74 BACE1 (0.59) SMN1; SMN2NOS1BACE1HSD17B10ALDH1A1
SCHEMBL965758 0.74
SCHEMBL12862676 0.74 SMN1; SMN2 (0.46) SMN1; SMN2NOS1BACE1HSD17B10GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0232623-B1 1-CARBACEPHALOSPORIN ANTIBIOTICS ELI LILLY AND COMPANY (US) 1993-03-17 EP disclosed
US-4892942-A 1-CARBA (DETHIA)CEPHALOSPORINS ELI LILLY AND COMPANY (US) 1990-01-09 US disclosed
US-4791106-A 1-Carbacephalosporin antibiotics ELI LILLY AND COMPANY (US) 1988-12-13 US disclosed
EP-0232623-A1 1-Carbacephalosporin antibiotics ELI LILLY AND COMPANY (US) 1987-08-19 EP disclosed