SCHEMBL9601313

SCHEMBL9601313

O=c1[nH]cc2ncc3ccccc3n12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 2/20 0.36
MAPK8 P45983 1/20 0.36
DYRK1A Q13627 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
CHEK1 O14757 1/20 0.35
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
DAO P14920 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
GMNN O75496 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33
NFKB1 P19838 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29354440 0.71 SMN1; SMN2 (0.39) DAOSMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL4510784 0.71 SMN1; SMN2 (0.39) DAOSMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL7854645 0.70 CA12 (0.40) CLK4MAPK8DYRK1ADYRK1BDAO
SCHEMBL7740296 0.67 DAO (0.34) CLK4MAPK8DYRK1ADYRK1BCHEK1
SCHEMBL9601750 0.67 KDM4E (0.46) CLK4MAPK8DYRK1ADYRK1BDAO
SCHEMBL7613241 0.66 KDM4E (0.43) DAOKDM4EALDH1A1HPGDMAPK1
SCHEMBL1602164 0.66 CHEK1 (0.54) CHEK1SMN1; SMN2L3MBTL1PBRM1PDE3B
SCHEMBL29881244 0.62 NPSR1 (0.47) DYRK1AKDM4EALDH1A1MAPTHPGD
SCHEMBL8229991 0.62 CA12 (0.52) DAOSMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL30692889 0.62 CA12 (0.52) DAOSMN1; SMN2KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993012113-A1 3-SUBSTITUTED IMIDAZO (1,5-a) AND IMIDAZO (1,5-a)-TRIAZOLO (1,5-c) QUINOXALINES AND QUINAZOLINES WITH CNS ACTIVITY THE UPJOHN COMPANY (US) 1993-06-24 WO disclosed