SCHEMBL9602297

SCHEMBL9602297

COc1nc2ccccc2c2c1ncn2C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.46
IKBKB O14920 5/20 0.44
CHUK O15111 5/20 0.44
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
POLB P06746 2/20 0.42
PDE4D Q08499 2/20 0.40
TLR7 Q9NYK1 2/20 0.40
LMNA P02545 1/20 0.40
HRH2 P25021 1/20 0.40
ADRA1D P25100 1/20 0.40
HTR2A P28223 1/20 0.40
ADORA2A P29274 1/20 0.40
ADRA1A P35348 1/20 0.40
NUDT1 P36639 1/20 0.40
HTR2B P41595 1/20 0.40
KCNH2 Q12809 1/20 0.40
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9218507 0.78 IKBKB (0.46) IKBKBCHUKPOLBPDE4DTLR7
SCHEMBL9601821 0.78 IKBKB (0.46) IKBKBCHUKHRH4POLBPDE4D
SCHEMBL3183969 0.78 TLR7 (0.62) ADORA3IKBKBCHUKPOLBPDE4D
SCHEMBL9603098 0.78 HTT (0.53) ADORA3MEN1KMT2ALMNAADORA2A
SCHEMBL9603118 0.78 TLR7 (0.69) ADORA3MEN1KMT2APOLBPDE4D
SCHEMBL9603045 0.76 IKBKB (0.72) IKBKBCHUK
SCHEMBL9602302 0.76 IKBKB (0.44) IKBKBCHUKMEN1KMT2APOLB
SCHEMBL30528123 0.75 IKBKB (0.46) IKBKBCHUKHRH4POLBPDE4D
SCHEMBL9602134 0.74 TLR7 (0.51) ADORA3POLBPDE4DTLR7LMNA
SCHEMBL9603056 0.74 HRH4 (0.47) IKBKBCHUKMEN1KMT2AHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4698348-A 1H-imidazo[4,5-c]quinolines and their use as bronchodilating agents RIKER LABORATORIES, INC. (US) 1987-10-06 US claimed
EP-0310950-B1 Quinoline intermediates for the synthesis of 1H-imidazo[4,5-c]quinolines and 1H-imidazo[4,5-c]quinolin-4-amimes RIKER LABORATORIES, INC. (US) 1993-01-13 EP disclosed
EP-0145340-B1 1H-Imidazo[4,5-c]quinolines and 1H-imidazo[4,5-c]quinolin-4-amines RIKER LABORATORIES, INC. (US) 1990-01-24 EP disclosed
EP-0310950-A1 Quinoline intermediates for the synthesis of 1H-imidazo[4,5-c]quinolines and 1H-imidazo[4,5-c]quinolin-4-amimes RIKER LABORATORIES, INC. (US) 1989-04-12 EP disclosed
US-4698348-A 1H-imidazo[4,5-c]quinolines and their use as bronchodilating agents RIKER LABORATORIES, INC. (US) 1987-10-06 US disclosed
EP-0145340-A2 1H-Imidazo[4,5-c]quinolines and 1H-imidazo[4,5-c]quinolin-4-amines RIKER LABORATORIES, INC. (US) 1985-06-19 EP disclosed