SCHEMBL9602503

SCHEMBL9602503

CC(Cc1cc2ccccc2s1)NO

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.54
ADRB2 P07550 1/20 0.54
ASIC3 Q9UHC3 1/20 0.50
LOXL2 Q9Y4K0 1/20 0.50
AGXT P21549 1/20 0.46
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
MMP1 P03956 1/20 0.42
FCER2 P06734 1/20 0.42
ALOX5 P09917 3/20 0.41
CYP1A2 P05177 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5962350 0.81 CYP2A6 (0.58) CYP2A6ADRB2ASIC3LOXL2AGXT
SCHEMBL30905568 0.78 CYP2A6 (0.59) CYP2A6ADRB2ASIC3LOXL2AGXT
SCHEMBL19760753 0.78 CYP2A6 (0.59) CYP2A6ADRB2ASIC3LOXL2AGXT
SCHEMBL20912808 0.78 CYP2A6 (0.59) CYP2A6ADRB2ASIC3LOXL2AGXT
SCHEMBL6637521 0.78 CYP2A6 (0.59) CYP2A6ADRB2ASIC3LOXL2AGXT
SCHEMBL5540703 0.78 CYP2A6 (0.55) CYP2A6ADRB2ASIC3LOXL2AGXT
SCHEMBL3459782 0.78 CYP2A6 (0.59) CYP2A6ADRB2ASIC3LOXL2AGXT
SCHEMBL18330737 0.77 CYP2A6 (0.47) CYP2A6ADRB2ASIC3LOXL2AGXT
Hydrochloric Acid SCHEMBL28235220 0.76 CYP2A6 (0.61) CYP2A6ADRB2ASIC3LOXL2AGXT
SCHEMBL9602507 0.74 AGXT (0.58) CYP2A6ADRB2ASIC3LOXL2AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0279263-B1 INDOLE, BENZOFURAN, BENZOTHIOPHENE CONTAINING LIPOXYGENASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1993-08-04 EP disclosed
US-4873259-A Indole, benzofuran, benzothiophene containing lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1989-10-10 US disclosed
EP-0279263-A2 Indole, benzofuran, benzothiophene containing lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1988-08-24 EP disclosed