SCHEMBL9602507

SCHEMBL9602507

CC(Cc1cc2ccccc2s1)ON

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGXT P21549 1/20 0.58
CYP2A6 P11509 3/20 0.54
ASIC3 Q9UHC3 1/20 0.54
LOXL2 Q9Y4K0 1/20 0.54
ADRB2 P07550 1/20 0.50
ADRA1D P25100 2/20 0.42
ALOX5 P09917 3/20 0.41
CYP1A2 P05177 2/20 0.41
PTGES O14684 1/20 0.41
LMNA P02545 1/20 0.41
LTA4H P09960 1/20 0.41
GAA P10253 1/20 0.41
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41
ALOX5AP P20292 1/20 0.41
LOX P28300 1/20 0.41
EPHX2 P34913 1/20 0.41
PTGS2 P35354 1/20 0.41
LTB4R Q15722 1/20 0.41
TAS1R3 Q7RTX0 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6637521 0.81 CYP2A6 (0.59) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL19760753 0.81 CYP2A6 (0.59) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL20912808 0.81 CYP2A6 (0.59) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL30905568 0.81 CYP2A6 (0.59) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL3459782 0.81 CYP2A6 (0.59) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL5962350 0.81 CYP2A6 (0.58) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL5540703 0.78 CYP2A6 (0.55) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL9602503 0.74 CYP2A6 (0.54) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL13760611 0.73 AGXT (0.62) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL7031640 0.73 AGXT (0.49) AGXTCYP2A6ASIC3LOXL2ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0279263-B1 INDOLE, BENZOFURAN, BENZOTHIOPHENE CONTAINING LIPOXYGENASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1993-08-04 EP disclosed
US-4873259-A Indole, benzofuran, benzothiophene containing lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1989-10-10 US disclosed
EP-0279263-A2 Indole, benzofuran, benzothiophene containing lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1988-08-24 EP disclosed