SCHEMBL9602900

SCHEMBL9602900

CCOP(=O)(Cc1cc[n+]([O-])cc1)OCC

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
TSHR P16473 2/20 0.39
NPY5R Q15761 1/20 0.38
MAPT P10636 1/20 0.35
CCNT1 O60563 2/20 0.34
CDK9 P50750 2/20 0.34
PPARD Q03181 1/20 0.34
HTT P42858 1/20 0.34
EGFR P00533 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HDAC1 Q13547 1/20 0.33
KCNH2 Q12809 1/20 0.33
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2962216 0.83 PPARD (0.40) CYP3A4CYP2C19TSHRPPARDNPSR1
SCHEMBL3375825 0.82 TSHR (0.50) TSHRNPY5RMAPTCCNT1CDK9
SCHEMBL16062693 0.81 POLB (0.46) CYP2C19TSHRNPY5RMAPTCCNT1
SCHEMBL2493713 0.77 TSHR (0.44) TSHRNPY5RMAPTCCNT1CDK9
SCHEMBL366215 0.77 NPY5R (0.50) TSHRNPY5RMAPTCCNT1CDK9
SCHEMBL23822678 0.76 TSHR (0.43) TSHRNPY5RMAPTCCNT1CDK9
SCHEMBL914767 0.76 NPY5R (0.49) TSHRNPY5RMAPTCCNT1CDK9
SCHEMBL916329 0.76 NPY5R (0.49) TSHRNPY5RMAPTCCNT1CDK9
SCHEMBL915242 0.76 TSHR (0.43) CYP3A4TSHRNPY5RMAPTCCNT1
SCHEMBL25923558 0.76 TSHR (0.43) TSHRNPY5RMAPTCCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5217963-A Antiischemic, antiepileptic agent CIBA-GEIGY CORPORATION (US) 1993-06-08 US disclosed
US-5057506-A Anticonvulsants, antispasmodic and antischemic agents CIBA-GEIGY CORPORATION (US) 1991-10-15 US disclosed
EP-0203891-B1 CERTAIN PHOSPHONIC ACIDS AND DERIVATIVES CIBA-GEIGY AG (CH) 1991-05-15 EP disclosed
US-4906621-A Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade CIBA-GEIGY CORPORATION (US) 1990-03-06 US disclosed
US-4898854-A NERVOUS SYSTEM DISORDERS CIBA-GEIGY CORPORATION (US) 1990-02-06 US disclosed
EP-0203891-A2 Certain phosphonic acids and derivatives CIBA-GEIGY AG (CH) 1986-12-03 EP disclosed