SCHEMBL9606682

SCHEMBL9606682

Cc1cc(Cl)cc(C)c1CNC(=O)C1CCC(=O)N1C

nearest known ligand 0.89

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 20/20 0.89

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2576645 0.94 P2RX7 (1.00) P2RX7
SCHEMBL2576644 0.94 P2RX7 (1.00) P2RX7
SCHEMBL2584153 0.84 P2RX7 (1.00) P2RX7
SCHEMBL2584150 0.84 P2RX7 (1.00) P2RX7
SCHEMBL2575507 0.82 P2RX7 (1.00) P2RX7
SCHEMBL2575509 0.82 P2RX7 (1.00) P2RX7
SCHEMBL2581635 0.82 P2RX7 (0.83) P2RX7
SCHEMBL2581636 0.82 P2RX7 (0.83) P2RX7
SCHEMBL2581837 0.78 P2RX7 (1.00) P2RX7
SCHEMBL2582027 0.78 P2RX7 (1.00) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049478-B1 SUBSTITUTED N-PHENYLMETHYL -5-OXO-PROLINE-2-AMIDES AS P2X7-RECEPTOR ANTAGONISTS AND THEIR METHODS OF USE GLAXO GROUP LTD (GB) 2012-05-30 EP disclosed