SCHEMBL9612380

SCHEMBL9612380

N#Cc1cc(-c2c(F)c(F)c(-c3cccc4c3ccc3cc5ccccc5cc34)c(F)c2F)cc(C#N)c1N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.37
PIM1 P11309 2/20 0.37
ESR1 P03372 4/20 0.35
ESR2 Q92731 4/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
MYB P10242 1/20 0.32
CES1 P23141 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
KDM4E B2RXH2 1/20 0.32
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
ALDH1A1 P00352 1/20 0.31
HIF1A Q16665 1/20 0.31
CYP1B1 Q16678 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ALOX15 P16050 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
DHODH Q02127 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13985609 0.89 MCL1 (0.38) MCL1PIM1ESR1ESR2CYP11B1
SCHEMBL8780567 0.81 MCL1 (0.41) MCL1PIM1ESR1ESR2CYP11B1
SCHEMBL13249122 0.74 DHODH (0.34) MCL1ESR1ESR2CYP11B1CYP11B2
SCHEMBL16122068 0.71 MCL1 (0.50) MCL1PIM1ESR1ESR2CYP11B1
SCHEMBL8780578 0.71 ALDH1A1 (0.47) MYBCES1ALDH1A1HIF1ACYP1B1
SCHEMBL17197648 0.70 CA1 (0.40) PIM1ESR1ESR2CA1CA2
SCHEMBL2709174 0.70 CES1 (0.41) CES1KDM4EALDH1A1HIF1ACYP1B1
SCHEMBL2551156 0.70 ALDH1A1 (0.52) CES1KDM4EALDH1A1HIF1ACYP1B1
SCHEMBL2867534 0.68 ALDH1A1 (0.58) CES1KDM4EALDH1A1HIF1ACYP1B1
SCHEMBL5750401 0.68 CA1 (0.46) PIM1KDM4ECA1CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2148909-B1 BENZANTHRACENE DERIVATIVES FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2012-05-30 EP disclosed