SCHEMBL9613243

SCHEMBL9613243

COC(=O)C1(NC(C)=O)CCC1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.50
ALDH1A1 P00352 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NPSR1 Q6W5P4 1/20 0.41
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
MEN1 O00255 1/20 0.34
CYP3A4 P08684 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.32
CNR2 P34972 1/20 0.32
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14276911 0.91 MAPT (0.44) MAPTALDH1A1L3MBTL1NPSR1CYP4F2
SCHEMBL15166977 0.80 MAPT (0.38) MAPTALDH1A1L3MBTL1NPSR1HTT
SCHEMBL8950840 0.80 SMN1; SMN2 (0.40) MAPTALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL12905301 0.80 MAPT (0.45) MAPTALDH1A1L3MBTL1NPSR1HTT
SCHEMBL12323501 0.80 MAPT (0.45) MAPTALDH1A1L3MBTL1NPSR1CYP4F2
SCHEMBL14271660 0.79 HTT (0.33) MAPTHTT
Hydrochloric Acid SCHEMBL9234685 0.77 MAPT (0.43) MAPTALDH1A1L3MBTL1NPSR1
SCHEMBL16068213 0.77 MAPT (0.44) MAPTALDH1A1L3MBTL1NPSR1CYP4F2
SCHEMBL9613093 0.77 FFAR3 (0.40) ALDH1A1CNR2HTT
SCHEMBL8587408 0.77 MAPT (0.34) MAPTALDH1A1L3MBTL1NPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021038426-A1 SUBSTITUTED 1,3-PHENYL HETEROARYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-03-04 WO disclosed
EP-1727797-B1 PROCESS FOR CROSS COUPLING INDOLES BOEHRINGER INGELHEIM PHARMA (US) 2012-05-30 EP disclosed
US-7408076-B2 2-Bromoanaline and 2-chloroaniline compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-05 US disclosed
US-7408076-B2 2-Bromoanaline and 2-chloroaniline compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-05 US disclosed
US-7332614-B2 Process for cross coupling indoles BOEHRINGER INGELHEIM INTERNATIONAL, GMBH (DE) 2008-02-19 US disclosed
US-7332614-B2 Process for cross coupling indoles BOEHRINGER INGELHEIM INTERNATIONAL, GMBH (DE) 2008-02-19 US disclosed