SCHEMBL9616211

SCHEMBL9616211

Oc1c2ccccc2cc2cc(Cl)ccc12

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.50
PTPN22 Q9Y2R2 1/20 0.42
TRPM4 Q8TD43 1/20 0.42
AHR P35869 1/20 0.41
NQO2 P16083 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CASP6 P55212 1/20 0.41
NQO1 P15559 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
GLA P06280 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methane SCHEMBL7938126 0.86 CYP2A6 (0.48) CYP2A6PTPN22TRPM4NQO2L3MBTL1
SCHEMBL437148 0.82 PTPN22 (0.56) CYP2A6PTPN22TRPM4NQO2L3MBTL1
Methane SCHEMBL155047 0.80 PTPN22 (0.54) PTPN22TRPM4NQO2L3MBTL1CASP6
Hydrogen Sulfide SCHEMBL27992660 0.80 PTPN22 (0.54) CYP2A6PTPN22TRPM4NQO2L3MBTL1
SCHEMBL29180044 0.80 PTPN22 (0.54) CYP2A6PTPN22TRPM4NQO2L3MBTL1
Methane SCHEMBL2327641 0.80 PTPN22 (0.54) PTPN22TRPM4NQO2L3MBTL1CASP6
SCHEMBL15763550 0.80 CYP2A6 (0.50) CYP2A6AHRL3MBTL1KDM4EMEN1
SCHEMBL18517084 0.80 CYP2A6 (0.50) CYP2A6AHRL3MBTL1ALDH1A1CYP1A2
SCHEMBL14743755 0.79 CYP1A2 (0.54) PTPN22TRPM4AHRNQO2CASP6
SCHEMBL29566119 0.79 AHR (0.47) CYP2A6AHRKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0416038-A4 NOVEL CHEMILUMINESCENT FUSED POLYCYCLIC RING-CONTAINING 1,2-DIOXETANES AND ASSAYS IN WHICH THEY ARE USED 1992-02-26 EP disclosed
EP-0416038-A1 NOVEL CHEMILUMINESCENT FUSED POLYCYCLIC RING-CONTAINING 1,2-DIOXETANES AND ASSAYS IN WHICH THEY ARE USED. TROPIX INC (US) 1991-03-13 EP disclosed
WO-1990000164-A1 NOVEL CHEMILUMINESCENT FUSED POLYCYCLIC RING-CONTAINING 1,2-DIOXETANES AND ASSAYS IN WHICH THEY ARE USED TROPIX, INC. (US) 1990-01-11 WO disclosed