SCHEMBL9616971

SCHEMBL9616971

CCCCCc1ccc(-c2nncs2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.56
RAB9A P51151 2/20 0.56
AKT1 P31749 7/20 0.52
PDPK1 O15530 1/20 0.52
ABCB11 O95342 1/20 0.52
AKT2 P31751 1/20 0.52
GAB1 Q13480 1/20 0.52
AKT3 Q9Y243 1/20 0.52
HSD11B1 P28845 1/20 0.49
HSD17B10 Q99714 3/20 0.45
ALDH1A1 P00352 3/20 0.45
MEN1 O00255 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
USP2 O75604 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
RARB P10826 5/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9616806 0.98 KDM4E (0.55) KDM4ERAB9AAKT1PDPK1ABCB11
SCHEMBL10589216 0.82 AKT1 (0.42) KDM4ERAB9AAKT1PDPK1ABCB11
SCHEMBL10162230 0.80 NPC1 (0.45) RAB9AAKT1MEN1MAPTKMT2A
SCHEMBL8742612 0.79 KDM4E (0.78) KDM4ERAB9AHSD11B1HSD17B10ALDH1A1
SCHEMBL9566995 0.78 RAB9A (0.54) KDM4ERAB9AALDH1A1MAPTHPGD
SCHEMBL9566994 0.78 RAB9A (0.54) KDM4ERAB9AALDH1A1MAPTHPGD
SCHEMBL10589213 0.78 PTPN11 (0.44) KDM4ERAB9AAKT1PDPK1ABCB11
SCHEMBL15164269 0.77 KDM4E (0.76) KDM4ERAB9AHSD11B1HSD17B10ALDH1A1
SCHEMBL15164268 0.77 KDM4E (0.76) KDM4ERAB9AHSD11B1HSD17B10ALDH1A1
SCHEMBL8742541 0.77 KDM4E (0.76) KDM4ERAB9AHSD11B1HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0309514-B1 MEDIA CONTAINING DERIVATIVES OF THIAZOLE AND THIADIAZOLE, WITH SMECTIC LIQUID-CRYSTAL PHASE MERCK PATENT GmbH (DE) 1992-12-02 EP disclosed
EP-0309514-A1 MEDIA CONTAINING DERIVATIVES OF THIAZOLE AND THIADIAZOLE, WITH SMECTIC LIQUID-CRYSTAL PHASE. MERCK PATENT GMBH (DE) 1989-04-05 EP disclosed
WO-1988008019-A1 MEDIA CONTAINING DERIVATIVES OF THIAZOLE AND THIADIAZOLE, WITH SMECTIC LIQUID-CRYSTAL PHASE MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-10-20 WO disclosed