SCHEMBL9621005

SCHEMBL9621005

COc1cc2c(cc1OC)CCCC(C(=O)O)=C2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 2/20 0.41
GLA P06280 2/20 0.41
MAOA P21397 2/20 0.41
HSD17B10 Q99714 3/20 0.38
KMT2A Q03164 1/20 0.38
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA4 P22748 2/20 0.38
CA6 P23280 2/20 0.38
CA7 P43166 2/20 0.38
CA9 Q16790 2/20 0.38
CA14 Q9ULX7 2/20 0.38
TPMT P51580 1/20 0.38
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.37
BRD4 O60885 1/20 0.37
LCK P06239 1/20 0.37
FYN P06241 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10448152 0.98 KDM4E (0.40) KDM4EALDH1A1GLAMAOAHSD17B10
SCHEMBL9621100 0.97 KDM4E (0.41) KDM4EALDH1A1GLAMAOAHSD17B10
SCHEMBL9621103 0.97 KDM4E (0.41) KDM4EALDH1A1GLAMAOAHSD17B10
SCHEMBL1589841 0.90 KDM4E (0.42) KDM4EALDH1A1GLAMAOAHSD17B10
SCHEMBL9620994 0.86 KDM4E (0.40) KDM4EALDH1A1GLAMAOAHSD17B10
SCHEMBL9621327 0.85 CHRNA7 (0.49) KMT2ASMN1; SMN2
SCHEMBL9621006 0.85 CHRNA7 (0.49) KMT2ASMN1; SMN2
SCHEMBL9620678 0.84 TSHR (0.41) ALDH1A1HSD17B10KMT2ACYP3A4MAPT
SCHEMBL9620925 0.83 KDM4E (0.40) KDM4EALDH1A1GLAMAOAHSD17B10
SCHEMBL9620921 0.83 KDM4E (0.40) KDM4EALDH1A1GLAMAOAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0284359-B1 1,4-DISUBSTITUTED PIPERAZINE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1992-01-08 EP disclosed
EP-0425134-A1 Condensed pyrrolo derivatives, process for their preparation and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1991-05-02 EP disclosed
US-4880809-A HYPOTENSIVE AGENTS, AMIDE DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-11-14 US disclosed
EP-0284359-A1 1,4-Disubstituted piperazine compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1988-09-28 EP disclosed