SCHEMBL9621100

SCHEMBL9621100

COc1cc2c(cc1OC)CCCC/C(C(=O)O)=C\2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 3/20 0.41
GLA P06280 2/20 0.41
MAOA P21397 2/20 0.41
HTT P42858 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 3/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA7 P43166 1/20 0.38
TPMT P51580 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
MAPT P10636 3/20 0.37
CYP3A4 P08684 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9621103 1.00 KDM4E (0.41) KDM4EALDH1A1GLAMAOAHTT
SCHEMBL9621005 0.97 KDM4E (0.41) KDM4EALDH1A1GLAMAOAHTT
Hydrochloric Acid SCHEMBL10448152 0.95 KDM4E (0.40) KDM4EALDH1A1GLAMAOAHTT
SCHEMBL1589841 0.90 KDM4E (0.42) KDM4EALDH1A1GLAMAOAHSD17B10
SCHEMBL9620921 0.86 KDM4E (0.40) KDM4EALDH1A1GLAMAOAHTT
SCHEMBL9620925 0.86 KDM4E (0.40) KDM4EALDH1A1GLAMAOAHTT
SCHEMBL9620994 0.83 KDM4E (0.40) KDM4EALDH1A1GLAMAOAHTT
SCHEMBL9621006 0.83 CHRNA7 (0.49) KMT2ASMN1; SMN2HPGDRAB9AMEN1
SCHEMBL9621327 0.83 CHRNA7 (0.49) KMT2ASMN1; SMN2HPGDRAB9AMEN1
SCHEMBL1590323 0.82 CYP3A4 (0.45) KDM4EALDH1A1GLAMAOAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0284359-B1 1,4-DISUBSTITUTED PIPERAZINE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1992-01-08 EP disclosed
US-4880809-A HYPOTENSIVE AGENTS, AMIDE DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-11-14 US disclosed
EP-0284359-A1 1,4-Disubstituted piperazine compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1988-09-28 EP disclosed