SCHEMBL9621206

SCHEMBL9621206

NC(=O)Nn1cnc2c(N)ncnc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.50
ADORA2A P29274 7/20 0.49
ADORA1 P30542 4/20 0.49
ADCY5 O95622 3/20 0.47
ALDH1A1 P00352 1/20 0.47
AHCY P23526 2/20 0.46
PI4KA P42356 3/20 0.45
PI4K2B Q8TCG2 3/20 0.45
PI4K2A Q9BTU6 3/20 0.45
PI4KB Q9UBF8 3/20 0.45
ADORA2B P29275 2/20 0.45
HSP90B1 P14625 1/20 0.45
EGFR P00533 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
NFKB1 P19838 1/20 0.44
THPO P40225 1/20 0.44
BLM P54132 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28210687 0.86 ADORA2A (0.51) GSK3BADORA2AADORA1ADCY5ALDH1A1
SCHEMBL28601746 0.84 ADORA2A (0.49) GSK3BADORA2AADORA1AHCYPI4KA
SCHEMBL22399264 0.78 ADORA2A (0.56) ADORA2AADORA1AHCYPI4KAPI4K2B
SCHEMBL9120 0.76 ADORA2A (0.59) ADORA2AADORA1AHCYPI4KAPI4K2B
SCHEMBL48453 0.75 ADORA2A (0.50) GSK3BADORA2AADORA1AHCYPI4KA
SCHEMBL7278433 0.75 ALDH1A1 (0.51) GSK3BADORA2AADORA1ADCY5ALDH1A1
SCHEMBL7278435 0.75 ALDH1A1 (0.51) GSK3BADORA2AADORA1ADCY5ALDH1A1
SCHEMBL3802976 0.75 EGFR (0.61) GSK3BPI4KAPI4K2BPI4K2API4KB
SCHEMBL2346678 0.75 GSK3B (0.67) GSK3BADORA2AADORA1ADCY5ALDH1A1
SCHEMBL20208091 0.73 ADORA2A (0.56) ADORA2AADORA1AHCYPI4KAPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0186454-B1 6-PURINYL N-(2-CHLOROETHYL) CARBAMATE AND THIOCARBAMATE, A PROCESS FOR THEIR PREPARATION AND USE THEREOF SPOFA Spojené Podniky Pro Zdravotnickou Vyrobu (CS) 1992-04-08 EP disclosed
US-4720497-A 6-purinyl N-/2-chloroethyl/carbamate and thiocarbamate and process for the preparation thereof SPOFA, SPOJENE PODNIKY PRO ZDRAVOTNICKOU VYROBU (CS) 1988-01-19 US disclosed
EP-0186454-A2 6-Purinyl N-(2-chloroethyl) carbamate and thiocarbamate, a process for their preparation and use thereof SPOFA Spojené Podniky Pro Zdravotnickou Vyrobu (CS) 1986-07-02 EP disclosed