SCHEMBL9623554

SCHEMBL9623554

COC(=O)CCc1[nH]cnc1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.40
KMT2A Q03164 2/20 0.38
GAA P10253 2/20 0.38
MEN1 O00255 1/20 0.38
ALOX12 P18054 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 2/20 0.37
HSD17B10 Q99714 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HPGD P15428 2/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
MAPK1 P28482 2/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
KDM5B Q9UGL1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3588654 0.83 KDM4E (0.43) TSHRGAAKDM4EALDH1A1HSD17B10
SCHEMBL6930989 0.82 EGFR (0.39) TSHRKMT2AKDM4EALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL3588652 0.81 KDM4E (0.43) TSHRGAAKDM4EALDH1A1HSD17B10
SCHEMBL1311876 0.81 HSD17B10 (0.44) GAANPSR1KDM4EHSD17B10
SCHEMBL1311858 0.79 CYP2C19 (0.36) TSHRKDM4EHSD17B10TDP1
Hydrochloric Acid SCHEMBL1311861 0.79 HSD17B10 (0.43) GAANPSR1KDM4EHSD17B10
SCHEMBL8891350 0.77 GABRR1 (0.53) KDM4EALDH1A1HSD17B10SMN1; SMN2HPGD
SCHEMBL16064995 0.73 QPCT (0.51) TSHRKMT2AMEN1NPSR1KDM4E
SCHEMBL5157739 0.72
SCHEMBL12844533 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5140034-A Hydroxytryptamine receptor antagonists; psychological and gastrointestinal disorders MERCK SHARP & DOHME LTD. (GB) 1992-08-18 US disclosed