SCHEMBL9624901

SCHEMBL9624901

COc1cc2c(cc1OC)C(=O)N(CCCN(C)CCc1csc3ccc(Br)cc13)C2

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 2/20 0.43
MAPT P10636 2/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
SMPD1 P17405 4/20 0.37
CHRM2 P08172 1/20 0.35
HTR1A P08908 1/20 0.35
SLC6A4 P31645 1/20 0.35
DRD3 P35462 1/20 0.35
KCNH2 Q12809 1/20 0.35
CYP2A6 P11509 1/20 0.35
ABCB1 P08183 2/20 0.35
MAOA P21397 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624336 0.90 MAPT (0.44) HCN4MAPTCYP3A4ALOX15SMPD1
SCHEMBL9624202 0.90 HCN4 (0.44) HCN4MAPTCYP3A4ALOX15SMPD1
SCHEMBL9624219 0.89 MAPT (0.45) HCN4MAPTCYP3A4ALOX15SMPD1
SCHEMBL9624311 0.89 CYP2A6 (0.37) HCN4MAPTCYP3A4ALOX15CYP2A6
Hydrochloric Acid SCHEMBL9624526 0.88 CYP3A4 (0.46) HCN4MAPTCYP3A4ALOX15SMPD1
SCHEMBL9623739 0.86 CYP2A6 (0.35) HCN4MAPTCYP3A4ALOX15CYP2A6
SCHEMBL9624113 0.85 HCN4 (0.44) HCN4MAPTCYP3A4ALOX15SMPD1
SCHEMBL9623834 0.85 HCN4 (0.43) HCN4MAPTCYP3A4ALOX15SMPD1
SCHEMBL10670769 0.85 HCN4 (0.64) HCN4MAPTCYP3A4ALOX15SMPD1
SCHEMBL9624996 0.84 MAPT (0.42) HCN4MAPTCYP3A4ALOX15SMPD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed