SCHEMBL9623739

SCHEMBL9623739

CN(CCCN1Cc2cc3c(cc2C1=O)OCO3)CCc1csc2ccc(Br)cc12

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.35
MAPT P10636 4/20 0.33
CA2 P00918 1/20 0.33
TP53 P04637 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
HCN4 Q9Y3Q4 1/20 0.31
CYP3A4 P08684 1/20 0.30
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624301 0.90 MAPT (0.35) MAPTCA2TP53HCN4CYP3A4
SCHEMBL9625186 0.89 SMPD1 (0.34) MAPTHCN4
SCHEMBL9624311 0.89 CYP2A6 (0.37) CYP2A6MAPTCA2TP53SIGMAR1
SCHEMBL9624641 0.88 MTNR1A (0.39) MAPTHCN4CYP3A4ALOX15
SCHEMBL9624901 0.86 HCN4 (0.43) CYP2A6MAPTHCN4CYP3A4ALOX15
SCHEMBL9624076 0.85 PRKCB (0.33) MAPT
SCHEMBL9624436 0.84 PRKCB (0.33)
SCHEMBL9623564 0.83 SMPD1 (0.36) MAPTHCN4CYP3A4ALOX15
SCHEMBL9625146 0.83 SLC6A4 (0.46) SIGMAR1
SCHEMBL9624428 0.82 KDM4E (0.32) MAPTHCN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed