SCHEMBL9624977

SCHEMBL9624977

COc1cc2c(cc1OC)CN(CCCN(C)CCCc1cccnc1)CC2

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 12/20 0.54
ABCG2 Q9UNQ0 1/20 0.54
DHCR7 Q9UBM7 2/20 0.46
TMEM97 Q5BJF2 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
HCRTR2 O43614 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624421 0.96 ABCB1 (0.54) ABCB1ABCG2DHCR7TMEM97SIGMAR1
SCHEMBL9624273 0.89 SIGMAR1 (0.42) ABCB1ABCG2SIGMAR1
SCHEMBL9624542 0.89 SMPD1 (0.46) ABCB1ABCG2SIGMAR1HCRTR2
SCHEMBL9624683 0.88 ABCB1 (0.55) ABCB1ABCG2DHCR7
SCHEMBL9623814 0.85 SIGMAR1 (0.41) ABCB1ABCG2SIGMAR1
SCHEMBL9624715 0.85 SIGMAR1 (0.45) ABCB1ABCG2SIGMAR1
SCHEMBL9625255 0.81 SIGMAR1 (0.45) ABCB1ABCG2SIGMAR1
SCHEMBL9625044 0.81 HCN4 (0.52) ABCB1
SCHEMBL10521178 0.81 ABCB1 (0.55) ABCB1ABCG2DHCR7SIGMAR1
SCHEMBL9624549 0.81 CHRNA7 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed