SCHEMBL9626233

SCHEMBL9626233

CC1(n2cc(C(=O)O)c(=O)c3cc(F)c(N4CCNCC4)cc32)CC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.68
KDM4E B2RXH2 6/20 0.68
LMNA P02545 6/20 0.68
HSD17B10 Q99714 5/20 0.68
HPGD P15428 5/20 0.68
BRD4 O60885 1/20 0.68
TSHR P16473 1/20 0.68
HTT P42858 1/20 0.68
CYP2J2 P51589 1/20 0.68
NPSR1 Q6W5P4 1/20 0.68
CYP2C9 P11712 2/20 0.65
CYP1A2 P05177 1/20 0.65
TOP2A P11388 1/20 0.65
TOP2B Q02880 1/20 0.65
DRD3 P35462 1/20 0.53
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
MAPT P10636 1/20 0.49
NPC1 O15118 1/20 0.48
ATP6V1B2 P21281 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10745959 0.88 ALDH1A1 (0.67) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL22372463 0.88 ALDH1A1 (0.65) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL9008319 0.88 ALDH1A1 (0.65) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL10748665 0.87 ALDH1A1 (0.53) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL9626236 0.87 ALDH1A1 (0.54) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL5083273 0.84 ALDH1A1 (0.67) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL11392814 0.84 ALDH1A1 (0.74) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL30605634 0.84 ALDH1A1 (0.74) ALDH1A1KDM4ELMNAHSD17B10HPGD
Hydrochloric Acid SCHEMBL11026221 0.83 ALDH1A1 (0.73) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL13916906 0.82 ALDH1A1 (0.46) ALDH1A1KDM4ELMNAHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4705788-A Novel antibacterial 7-amino-1(substituted cyclopropyl)-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids BAYER AKTIENGESELLSCHAFT (DE) 1987-11-10 US claimed
EP-0198192-B1 7-AMINO-1-(SUBST.CYCLOPROPYL)-1,4 -DIHYDRO-4-OXO-QUINOLINE CARBOXYLIC ACIDS, METHOD FOR THEIR PREPARATION, AND ANTIBACTERIAL AGENTS CONTAINING THEM BAYER AG (DE) 1992-05-13 EP disclosed
EP-0300155-A2 Cyclopropyl amines BAYER AG (DE) 1989-01-25 EP disclosed
US-4705788-A Novel antibacterial 7-amino-1(substituted cyclopropyl)-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids BAYER AKTIENGESELLSCHAFT (DE) 1987-11-10 US disclosed
EP-0198192-A1 7-Amino-1-(subst.cyclopropyl)-1,4 -dihydro-4-oxo-quinoline carboxylic acids, method for their preparation, and antibacterial agents containing them BAYER AG (DE) 1986-10-22 EP disclosed