SCHEMBL9628683

SCHEMBL9628683

CCCN(CCC)C(=O)c1cc2cc([N+](=O)[O-])ccc2s1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.81
HPGD P15428 2/20 0.81
CYP1A2 P05177 1/20 0.81
CYP2C9 P11712 1/20 0.81
CYP2C19 P33261 1/20 0.81
POLB P06746 4/20 0.62
LMNA P02545 4/20 0.55
SMN1; SMN2 Q16637 4/20 0.55
ALDH1A1 P00352 2/20 0.51
GAA P10253 2/20 0.49
RAB9A P51151 4/20 0.48
TDP1 Q9NUW8 3/20 0.46
NPC1 O15118 2/20 0.46
MAPT P10636 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPK1 P28482 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.43
HDAC3 O15379 2/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC2 Q92769 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6233545 0.82 KMT2A (0.73) KMT2AHPGDCYP1A2CYP2C9CYP2C19
SCHEMBL9627805 0.81 KMT2A (0.53) KMT2AHPGDCYP1A2CYP2C9CYP2C19
SCHEMBL9486762 0.80 POLB (0.67) KMT2AHPGDCYP1A2CYP2C9CYP2C19
SCHEMBL2977014 0.78 SMN1; SMN2 (0.66) KMT2AHPGDCYP1A2CYP2C9CYP2C19
SCHEMBL23612325 0.76 POLB (0.61) KMT2AHPGDCYP1A2CYP2C9CYP2C19
SCHEMBL1000630 0.76 KMT2A (0.64) KMT2AHPGDCYP1A2CYP2C9CYP2C19
SCHEMBL1491507 0.76 POLB (0.63) KMT2AHPGDCYP1A2CYP2C9CYP2C19
SCHEMBL9628692 0.75 MAPK1 (0.47) KMT2AHPGDCYP1A2CYP2C9CYP2C19
SCHEMBL5439326 0.75 SMN1; SMN2 (0.62) KMT2AHPGDCYP1A2CYP2C9CYP2C19
SCHEMBL312150 0.75 POLB (0.66) KMT2AHPGDCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP disclosed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP disclosed