SCHEMBL9628909

SCHEMBL9628909

COC(=O)C(c1ccccc1)c1ccc(OCC(O)CNC(C)C)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.67
ADRB1 P08588 4/20 0.67
CYP2D6 P10635 2/20 0.67
ADRB3 P13945 2/20 0.67
KMT2A Q03164 3/20 0.59
MEN1 O00255 2/20 0.59
PTGS1 P23219 1/20 0.58
SLC6A2 P23975 1/20 0.58
CYP1A2 P05177 2/20 0.57
TSHR P16473 2/20 0.57
OPRK1 P41145 1/20 0.57
ALOX15 P16050 1/20 0.57
CYP2C19 P33261 1/20 0.57
TDP1 Q9NUW8 3/20 0.56
LMNA P02545 2/20 0.56
PMP22 Q01453 2/20 0.56
CNR1 P21554 1/20 0.56
ADRA1D P25100 1/20 0.56
ADRA1A P35348 1/20 0.56
ADRA1B P35368 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28473884 0.84 MAPT (0.63) ADRB2ADRB1CYP2D6ADRB3KMT2A
SCHEMBL7367812 0.81 ADRB2 (1.00) ADRB2ADRB1CYP2D6ADRB3KMT2A
SCHEMBL8266174 0.81 ADRB2 (1.00) ADRB2ADRB1CYP2D6ADRB3KMT2A
SCHEMBL6672267 0.81 ADRB2 (0.67) ADRB2ADRB1CYP2D6ADRB3KMT2A
Hydrochloric Acid SCHEMBL10872169 0.80 ADRB2 (0.97) ADRB2ADRB1CYP2D6ADRB3KMT2A
Acetamide SCHEMBL5800005 0.79 ADRB2 (0.83) ADRB2ADRB1CYP2D6ADRB3KMT2A
SCHEMBL11232155 0.79 ADRB2 (0.88) ADRB2ADRB1CYP2D6ADRB3KMT2A
SCHEMBL11667770 0.79 ADRB2 (0.88) ADRB2ADRB1CYP2D6ADRB3PTGS1
SCHEMBL4455319 0.79 ADRB2 (0.63) ADRB2ADRB1CYP2D6ADRB3KMT2A
SCHEMBL11594087 0.79 ADRB2 (0.72) ADRB2ADRB1CYP2D6ADRB3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0256586-B1 PROCESS FOR THE PREPARATION OF ESTERS OF 4-(2,3-EPOXYPROPOXY)PHENYLACETIC ACID AND 4-(2-HYDROXY-3-ISOPROPYLAMINO-PROPOXY)PHENYLACETIC ACID AND/OR ATENOLOL IN STEREOSPECIFIC FORM GIST-BROCADES N.V. (NL) 1992-05-13 EP disclosed
EP-0256586-A1 Process for the preparation of esters of 4-(2,3-epoxypropoxy)phenylacetic acid and 4-(2-hydroxy-3-isopropylamino-propoxy)phenylacetic acid and/or atenolol in stereospecific form GIST-BROCADES N.V. (NL) 1988-02-24 EP disclosed