SCHEMBL9629256

SCHEMBL9629256

O=c1oc2ccccc2cc1CCN1CCC(Nc2nc3ccccc3n2Cc2cnccn2)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 15/20 0.46
EED O75530 2/20 0.45
SSTR5 P35346 3/20 0.43
NR4A2 P43354 1/20 0.42
DRD2 P14416 2/20 0.40
HTR2A P28223 2/20 0.40
HTR7 P34969 2/20 0.40
HTR6 P50406 2/20 0.40
MEN1 O00255 1/20 0.40
MLNR O43193 1/20 0.40
CACNA1F O60840 1/20 0.40
USP2 O75604 1/20 0.40
ABCB11 O95342 1/20 0.40
EGFR P00533 1/20 0.40
LMNA P02545 1/20 0.40
HLA-A P04439 1/20 0.40
ERBB2 P04626 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
LCK P06239 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1151833 0.87 KCNH2 (0.50) KCNH2EEDSSTR5NR4A2DRD2
Hydrochloric Acid SCHEMBL10857686 0.86 KCNH2 (0.51) KCNH2EEDSSTR5NR4A2DRD2
Water SCHEMBL1152258 0.84 KCNH2 (0.55) KCNH2EEDSSTR5NR4A2DRD2
SCHEMBL9631586 0.82 KCNH2 (0.50) KCNH2EEDSSTR5NR4A2DRD2
Hydrochloric Acid SCHEMBL1151990 0.82 KCNH2 (0.48) KCNH2EEDSSTR5NR4A2DRD2
Hydrochloric Acid SCHEMBL10428750 0.81 KCNH2 (0.49) KCNH2EEDSSTR5NR4A2DRD2
Oxalic Acid SCHEMBL9630385 0.81 SSTR5 (0.62) KCNH2EEDSSTR5NR4A2DRD2
Oxalic Acid SCHEMBL9630381 0.81 SSTR5 (0.62) KCNH2EEDSSTR5NR4A2DRD2
SCHEMBL1151704 0.80 KCNH2 (0.51) KCNH2EEDSSTR5NR4A2DRD2
SCHEMBL10428783 0.80 SSTR5 (0.70) KCNH2EEDSSTR5NR4A2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5151424-A Antiallergens or antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-29 US disclosed
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed
US-5071846-A Anti-hystaminic [(bicyclic heterocyclyl) methyl and --hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1991-12-10 US disclosed
US-4988689-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1991-01-29 US disclosed
EP-0297661-A1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1989-01-04 EP disclosed