SCHEMBL9629376

SCHEMBL9629376

c1csc(Cn2c(NC3CCNC3)nc3ccccc32)c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.57
NR4A2 P43354 2/20 0.57
SMN1; SMN2 Q16637 3/20 0.49
TSHR P16473 3/20 0.49
KDM4E B2RXH2 2/20 0.49
MAPT P10636 2/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
RAB9A P51151 1/20 0.44
HTT P42858 2/20 0.43
SSTR5 P35346 4/20 0.43
MAOB P27338 1/20 0.42
HTR6 P50406 1/20 0.42
ALOX15 P16050 1/20 0.42
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
CFTR P13569 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL9629446 0.94 KCNH2 (0.52) KCNH2NR4A2SMN1; SMN2TSHRKDM4E
SCHEMBL9698816 0.94 KCNH2 (0.65) KCNH2NR4A2SMN1; SMN2TSHRKDM4E
SCHEMBL9631535 0.85 MAPT (0.42) KCNH2NR4A2MAPTHPGDMAOB
Hydrochloric Acid SCHEMBL9631314 0.84 MAPT (0.42) KCNH2NR4A2MAPTHPGDMAOB
SCHEMBL7860383 0.81 KCNH2 (0.48) KCNH2NR4A2SMN1; SMN2TSHRKDM4E
SCHEMBL7860380 0.81 KCNH2 (0.48) KCNH2NR4A2SMN1; SMN2TSHRKDM4E
SCHEMBL9629886 0.80 KCNH2 (0.88) KCNH2NR4A2SMN1; SMN2MAPTHTT
Hydrochloric Acid SCHEMBL9630387 0.79 KCNH2 (0.57) KCNH2NR4A2TSHRKDM4EHTT
SCHEMBL9740847 0.78 SSTR5 (0.54) KCNH2NR4A2SMN1; SMN2TSHRKDM4E
Bromide SCHEMBL9630112 0.78 KCNH2 (0.54) KCNH2NR4A2MAPTSSTR5MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5151424-A Antiallergens or antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-29 US disclosed
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed
US-5071846-A Anti-hystaminic [(bicyclic heterocyclyl) methyl and --hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1991-12-10 US disclosed
US-4988689-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1991-01-29 US disclosed