Oxalic Acid

Oxalic Acid

SCHEMBL9629446

O=C(O)C(=O)O.c1csc(Cn2c(NC3CCNC3)nc3ccccc32)c1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.52
NR4A2 P43354 1/20 0.52
TSHR P16473 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
NPSR1 Q6W5P4 2/20 0.42
HTT P42858 2/20 0.42
SSTR5 P35346 2/20 0.41
OPRK1 P41145 1/20 0.41
MAOB P27338 1/20 0.40
HTR6 P50406 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
ITK Q08881 1/20 0.40
RAB9A P51151 1/20 0.40
CHEK2 O96017 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9629376 0.94 KCNH2 (0.57) KCNH2NR4A2TSHRSMN1; SMN2KDM4E
SCHEMBL9698816 0.88 KCNH2 (0.65) KCNH2NR4A2TSHRSMN1; SMN2KDM4E
Oxalic Acid SCHEMBL9630409 0.82 SSTR5 (0.45) KCNH2NR4A2TSHRSMN1; SMN2KDM4E
Oxalic Acid SCHEMBL9630418 0.82 SSTR5 (0.45) KCNH2NR4A2TSHRSMN1; SMN2KDM4E
SCHEMBL9631535 0.80 MAPT (0.42) KCNH2NR4A2MAPTHPGDMAOB
Hydrochloric Acid SCHEMBL9631314 0.79 MAPT (0.42) KCNH2NR4A2MAPTHPGDMAOB
SCHEMBL7860383 0.78 KCNH2 (0.48) KCNH2NR4A2TSHRSMN1; SMN2KDM4E
SCHEMBL7860380 0.78 KCNH2 (0.48) KCNH2NR4A2TSHRSMN1; SMN2KDM4E
SCHEMBL9698262 0.76 SMN1; SMN2 (0.54) TSHRSMN1; SMN2KDM4EMAPTHPGD
SCHEMBL9630499 0.75 SMN1; SMN2 (0.51) TSHRSMN1; SMN2KDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5151424-A Antiallergens or antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-29 US disclosed
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed
US-5071846-A Anti-hystaminic [(bicyclic heterocyclyl) methyl and --hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1991-12-10 US disclosed
US-4988689-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1991-01-29 US disclosed
EP-0297661-A1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1989-01-04 EP disclosed