SCHEMBL9629561

SCHEMBL9629561

CC(=O)Oc1ccc(OC[C@@H](O)CNC(C)C)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.71
ADRB1 P08588 4/20 0.71
CYP2D6 P10635 3/20 0.71
ADRB3 P13945 2/20 0.71
CYP1A2 P05177 2/20 0.71
TSHR P16473 2/20 0.71
OPRK1 P41145 1/20 0.71
MEN1 O00255 1/20 0.71
ALOX15 P16050 1/20 0.71
CYP2C19 P33261 1/20 0.71
KMT2A Q03164 1/20 0.71
PTGS1 P23219 1/20 0.68
SLC6A2 P23975 1/20 0.68
LMNA P02545 2/20 0.65
TDP1 Q9NUW8 2/20 0.65
CNR1 P21554 1/20 0.65
ADRA1D P25100 1/20 0.65
ADRA1A P35348 1/20 0.65
ADRA1B P35368 1/20 0.65
KDM4E B2RXH2 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9629567 1.00 ADRB2 (0.71) ADRB2ADRB1CYP2D6ADRB3CYP1A2
SCHEMBL11594190 0.90 PTGS1 (0.67) ADRB2ADRB1CYP2D6ADRB3CYP1A2
SCHEMBL10614283 0.87 ADRB2 (0.56) ADRB2ADRB1CYP2D6ADRB3CYP1A2
SCHEMBL11251793 0.86 PTGS1 (0.65) ADRB2ADRB1CYP2D6ADRB3CYP1A2
Hydrochloric Acid SCHEMBL11170713 0.85 MAPT (0.64) ADRB2ADRB1CYP2D6ADRB3CYP1A2
SCHEMBL11595152 0.85 PTGS1 (0.68) ADRB2ADRB1CYP2D6ADRB3CYP1A2
SCHEMBL11594087 0.83 ADRB2 (0.72) ADRB2ADRB1CYP2D6ADRB3CYP1A2
Practolol SCHEMBL39926 0.83 ADRB2 (1.00) ADRB2ADRB1CYP2D6ADRB3CYP1A2
Practolol SCHEMBL39925 0.83 ADRB2 (1.00) ADRB2ADRB1CYP2D6ADRB3CYP1A2
SCHEMBL10961494 0.83 ADRB2 (0.78) ADRB2ADRB1CYP2D6ADRB3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0256586-B1 PROCESS FOR THE PREPARATION OF ESTERS OF 4-(2,3-EPOXYPROPOXY)PHENYLACETIC ACID AND 4-(2-HYDROXY-3-ISOPROPYLAMINO-PROPOXY)PHENYLACETIC ACID AND/OR ATENOLOL IN STEREOSPECIFIC FORM GIST-BROCADES N.V. (NL) 1992-05-13 EP disclosed
EP-0256586-A1 Process for the preparation of esters of 4-(2,3-epoxypropoxy)phenylacetic acid and 4-(2-hydroxy-3-isopropylamino-propoxy)phenylacetic acid and/or atenolol in stereospecific form GIST-BROCADES N.V. (NL) 1988-02-24 EP disclosed