SCHEMBL9632708

SCHEMBL9632708

FC(F)=C(F)CCSc1nnc(-c2nnc(SCCC(F)=C(F)F)o2)o1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.40
KDM4E B2RXH2 2/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
MAPT P10636 2/20 0.40
TP53 P04637 2/20 0.40
THRB P10828 1/20 0.40
POLB P06746 2/20 0.39
HSD17B10 Q99714 1/20 0.38
KMT2A Q03164 1/20 0.38
MAPK1 P28482 1/20 0.37
NPC1 O15118 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
LMNA P02545 1/20 0.36
PTGS1 P23219 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HTT P42858 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9631769 0.91 PKM (0.42) GLAKDM4ESMN1; SMN2MAPTTP53
SCHEMBL9632583 0.87 GLA (0.41) GLAKDM4ESMN1; SMN2MAPTTP53
SCHEMBL10364612 0.83 MAPT (0.56) GLASMN1; SMN2MAPTTP53POLB
SCHEMBL9631728 0.83 APEX1 (0.37) GLAKDM4ESMN1; SMN2MAPTTP53
SCHEMBL10364759 0.82 HTT (0.55) GLAKDM4ESMN1; SMN2MAPTTP53
SCHEMBL10363894 0.82 MAPT (0.60) GLAKDM4ESMN1; SMN2MAPTTP53
SCHEMBL10435183 0.80 GLA (0.37) GLAKDM4ESMN1; SMN2MAPTTP53
SCHEMBL10435187 0.80 GLA (0.37) GLAKDM4ESMN1; SMN2MAPTTP53
SCHEMBL9633107 0.79 GLA (0.34) GLAKDM4ESMN1; SMN2MAPTTP53
SCHEMBL10364618 0.78 MAPT (0.53) SMN1; SMN2MAPTTP53THRBPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0364396-A1 Neumaticides and fungicides CIBA-GEIGY AG (CH) 1990-04-18 EP claimed
US-5162349-A Mercaptobis/1,3,4-oxa- and -thiadiazoles/ CIBA-GEIGY CORPORATION (US) 1992-11-10 US disclosed
EP-0364396-A1 Neumaticides and fungicides CIBA-GEIGY AG (CH) 1990-04-18 EP disclosed